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Trazadone Drug Name:  
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Indications
Dosages
Interactions
Precautions
Contraindications
Adverse Reactions
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Interactions:

Buspirone

  • Adverse Effect: An elevated SGPT (ALT) level  
  • Clinical Management: During concurrent therapy with trazodone and buspirone, monitor liver function closely.

    Carbamazepine

  • Adverse Effect: An increased risk of carbamazepine toxicity (ataxia, nystagmus, diplopia, headache, vomiting, apnea, seizures)  
  • Clinical Management: Monitor for symptoms of carbamazepine toxicity when trazodone is added to therapy. Serum carbamazepine levels should also be considered with the addition or discontinuation of Trazadone and dosage adjustments made accordingly.

    Fluoxetine

  • Adverse Effect: trazodone toxicity (sedation, dry mouth, urinary retention) or serotonin syndrome (hypertension, hyperthermia, myoclonus, mental status changes)  
  • Clinical Management: Due to the potential for impairment in trazodone metabolism, patients should be monitored for any signs of trazodone toxicity. Occasional dosage reductions of trazodone may be required.

    Fluphenazine

  • Adverse Effect: Hypotension  
  • Clinical Management: Monitor blood pressure, particularly in patients who might be sensitive to this effect. Advise patient to rise slowly from lying or sitting position.

    Haloperidol

  • Adverse Effect: An increase in plasma concentrations of m-chlorophenylpiperazine (m-CPP), the active metabolite of trazodone

    Thioridazine

  • Adverse Effect: Hypotension  
  • Clinical Management: Monitor blood pressure, particularly in patients who might be sensitive to this effect. Advise patient to rise slowly from lying or sitting position.

    Tramadol

  • Adverse Effect: CNS depression (sedation, lethargy, speech difficulties)  
  • Clinical Management: Use caution if tramadol is to be used concomitantly in patients receiving trazodone therapy. Monitor patients for signs of CNS depression (sedation, lethargy, speech difficulties) and adjust doses accordingly. The manufacturer recommends that reduced dosages of tramadol be used when it is coadministered with other CNS depressants.

    Trifluoperazine

  • Adverse Effect: Hypotension  
  • Clinical Management: Monitor blood pressure, particularly in patients who might be sensitive to this effect. Advise patient to rise slowly from lying or sitting position
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