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Acetazolamide Drug Name:  
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Interactions:

Aspirin

  • Adverse Effect: salicylate toxicity (vomiting, tachycardia, hyperpnea, mental confusion) or acetazolamide toxicity (fatigue, lethargy, somnolence, confusion, hyperchloremic metabolic acidosis)
  • Clinical Management: If used concurrently (especially in patients with renal dysfunction or receiving large doses of aspirin), monitor for salicylate toxicity.

    Digoxin

  • Adverse Effect: Digoxin toxicity (nausea, vomiting, arrhythmias)  
  • Clinical Management: If concurrent therapy is required, monitor the patients electrolytes carefully, particularly potassium, and assess the need for electrolyte (ie, potassium) replacement therapy.

    Lithium

  • Adverse Effect: Decreased lithium effectiveness or increased lithium concentrations
  • Clinical Management: Monitor therapeutic efficacy of lithium and serum lithium concentrations. Adjustments of the lithium dose may be necessary.

    Phenytoin

  • Adverse Effect: An increased risk of osteomalacia  
  • Clinical Management: If acetazolamide and phenytoin therapy are to be coadministered, monitor patients for early signs of osteomalacia. Treatment of osteomalacia includes withdrawal of acetazolamide and administration of vitamin D and phosphate.

    Quinidine

  • Adverse Effect: quinidine toxicity (ventricular arrhythmias, hypotension, aggravated CHF)
  • Clinical Management: If initiating, discontinuing, or changing the dose of acetazolamide in patients taking quinidine, monitor quinidine levels and adjust quinidine dose as required.
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